// Workers AI · dad joke modeWhat did CP 55,244 say to its friend? "You're a number one buddy.
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Chemical compound
Pharmaceutical compound
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| Formula | C26H42O3 |
| Molar mass | 402.619 g·mol−1 |
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CP 55,244 is a chemical compound which is a cannabinoid receptor agonist. It has analgesic effects and is used in scientific research. It is an extremely potent CB1 full agonist with a Ki of 0.21 nM, making it more potent than the commonly used full agonist HU-210.[1][2]
See also
[edit]References
[edit]- ↑ Melvin LS, Milne GM, Johnson MR, Wilken GH, Howlett AC (November 1995). "Structure-activity relationships defining the ACD-tricyclic cannabinoids: cannabinoid receptor binding and analgesic activity". Drug Design and Discovery. 13 (2): 155–66. PMID 8872458.
- ↑ Griffin G, Wray EJ, Martin BR, Abood ME (October 1999). "Cannabinoid agonists and antagonists discriminated by receptor binding in rat cerebellum". British Journal of Pharmacology. 128 (3): 684–8. doi:10.1038/sj.bjp.0702806. PMC 1571656. PMID 10516649.
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| Oneirogens (unknown mech.) |
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| Cannabinoids (CB1 agonists) |
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